PEG-MGF

PEG-MGF is a PEGylated synthetic analog of mechano growth factor (MGF), an IGF-1 splice variant produced locally in response to mechanical loading, engineered with polyethylene glycol attachment to extend its in vivo half-life from minutes to days. It is studied for skeletal muscle repair, hypertrophy, and satellite cell activation. Placed on FDA Category 2 list (September 29, 2023) as 'Mechano growth factor pegylated (PEG-MGF).'

Preliminary evidence FDA Category 2 Growth Factor

Written by WhatPeptide Editorial Team · Last updated 2026-03-17

FDA Category 2 — compounding availability may be limited.

Half-life

Approximately 24-72 hours (PEGylation-extended)

Dosage range

200-400 mcg subcutaneously 1-2x weekly (research context)

Administration

Subcutaneous injection

Research level

Preliminary

How PEG-MGF works

Mechano growth factor activates distinct intracellular pathways from systemic IGF-1, particularly stimulating muscle satellite cell proliferation through an Akt-independent mechanism that may involve the unique E-domain of the MGF splice variant. PEGylation prevents rapid enzymatic degradation, enabling sustained engagement with receptors in damaged muscle tissue following systemic or local injection. Rodent studies demonstrate enhanced muscle fiber cross-sectional area and accelerated recovery after eccentric exercise or injury.

Also known as: PEGylated Mechano Growth Factor, PEG-Mechano Growth Factor, Pegylated IGF-1Ec

Research relevance

Muscle Growth
Moderate relevance 70
Recovery & Healing
Moderate relevance 55

Side effects & safety

Limited human safety data Potential hypoglycemia Injection site reactions Tumor promotion risk (theoretical)

Contraindications

Active or prior malignancy
Pregnancy
Diabetic retinopathy

Consult a healthcare provider before use if any of these apply to you.

Key studies

FAQ

What is PEG-MGF? +
PEG-MGF is a PEGylated synthetic analog of mechano growth factor (MGF), an IGF-1 splice variant produced locally in response to mechanical loading, engineered with polyethylene glycol attachment to extend its in vivo half-life from minutes to days. It is studied for skeletal muscle repair, hypertrophy, and satellite cell activation. Placed on FDA Category 2 list (September 29, 2023) as 'Mechano growth factor pegylated (PEG-MGF).' Its mechanism of action is based on preliminary or early-stage research.
What is PEG-MGF researched for? +
PEG-MGF has the strongest research relevance for Muscle Growth, Recovery & Healing. Evidence is based on preliminary or early-stage research.
What are the side effects of PEG-MGF? +
Reported side effects include Limited human safety data, Potential hypoglycemia, Injection site reactions, Tumor promotion risk (theoretical). Key contraindications: Active or prior malignancy; Pregnancy; Diabetic retinopathy.
Is PEG-MGF FDA approved? +
PEG-MGF is classified as FDA Category 2, meaning compounding availability may be limited.
How is PEG-MGF administered? +
PEG-MGF is typically administered via subcutaneous route. Researched dosage range: 200-400 mcg subcutaneously 1-2x weekly (research context). Half-life: Approximately 24-72 hours (PEGylation-extended).

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